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268

抑制剂 & 化合物

69

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Cat. No. Product Name Target Signaling Pathways
T9103 BVDV-IN-1

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
BVDV-IN-1 是一种牛病毒性腹泻病毒 (BVDV) 的非核苷抑制剂 (NNI),EC50 为 1.8 μM。它直接与 BVDV RdRp 的疏水口袋结合,对耐 NNI 氨基硫脲 (TSC) 的 BVDV 具有抗病毒活性。
T15573 Inarigivir soproxil

SB9200

HCV Protease Microbiology/Virology; Proteases/Proteasome
Inarigivir soproxil (SB9200) 是一种先天免疫激动剂。 它还显示出针对耐药丙型肝炎病毒 (HCV) 变体的有效抗病毒活性。在基因型 1 HCV 复制子系统细胞中, HCV 1a/1b 的 EC50 为 2.2 和 1.0 μM。
T8625 5-Fluorocytidine

Antiviral Immunology/Inflammation
5-Fluorocytidine 具有抗病毒活性。
T67904 Antiviral agent

HBV Microbiology/Virology
Antiviral agent是一种具有抗乙型肝炎活性的噻唑烷。
T19849L 2-PADQZ hydrochloride

2-PADQZ hydrochloride (60547-97-9 Free base)

Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology
2-PADQZ hydrochloride 显示出抗病毒活性并靶向甲型流感病毒 RNA 启动子。
T67785 ABI-1968

ABI-1968具有抗病毒和抗肿瘤活性。
T26020 R 61837

R-61837,R61837

Antiviral Immunology/Inflammation
R 61837 是一种新型鼻病毒抑制剂,是一种取代的苯基哒嗪胺,具有抗病毒活性。
T16913 Sotirimod

R850,S-30594

Virus Protease Microbiology/Virology
Sotirimod(R850) 是一种新型免疫调节剂,具有抗肿瘤和抗病毒活性,可用于研究光化性角化病。
T67806 Rociclovir

Antiviral Immunology/Inflammation
Rociclovir 具有抗病毒活性,可用于治疗病毒感染。
T1118L Cefprozil

Cefprozilum,Cefprozilo,Cefzil,Brisoral,Cefprozil anhydrous

Antibacterial; Antibiotic Microbiology/Virology
Cefprozil (Cefzil) 是一种新型头孢菌素类抗生素,具有抗病毒活性,可用于研究免疫系统疾病。
T26914 BTA-9881

BTA9881,AZD9639,AZD-9639,BTA 9881,MEDI-564

RSV Microbiology/Virology
BTA-9881 是一种具有口服活性的新型 RSV 融合抑制剂,具有抗病毒活性,可用于研究呼吸道合胞病毒感染。
T67797 DDG-39

1-(2,3-dideoxy-2-fluoropentofuranosyl)cytosine

Antiviral; HBV; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
DDG-39 (1-(2,3-dideoxy-2-fluoropentofuranosyl)cytosine)具有抗病毒活性,在细胞培养中具有有效的选择性抗 HIV-1 和HBV 活性。平均抗病毒 IC50为0.61μM。
T25702 Levovirin

ICN 17261,L-Ribavirin,ICN-17261,ICN17261

Levovirin is a monocyclic L-nucleosides with type 1 cytokine-inducing activity. Levovirin is the L-enantiomer of Ribavirin. Levovirin has similar immunomodulatory activity but does not have direct antiviral activity or hemolytic anemia.
T80675 IM-250

Antiviral Immunology/Inflammation
IM-250 具有抗病毒活性,IC值为 25 nm - 100 nM。
T60014 SHEN26

Antiviral Immunology/Inflammation
SHEN26 具有抗病毒活性,可用于治疗病毒感染的研究。
TNU0442 2’-beta-C-Methyl inosine

2'-C-Methylinosine

Antiviral; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation
2’-beta-C-Methyl inosine (2'-C-Methylinosine) 是一种 HCV RNA聚合酶抑制剂,具有抗病毒活性,可用用于研究用于治疗丙型肝炎病毒感染。
T6367 Abacavir sulfate

Abacavir Hemisulfate,硫酸阿巴卡韦,1592U89,ABC sulfate,Ziagen

Apoptosis; HIV Protease; Reverse Transcriptase Apoptosis; Microbiology/Virology; Proteases/Proteasome
Abacavir sulfate (Ziagen) 是一种核苷类似物逆转录酶抑制剂,可用于 HIV 和 AIDS。
T1649 Tenofovir

替诺福韦,泰诺福韦,PMPA,TDF,GS 1278

HBV; HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Tenofovir (GS 1278) 是一种核苷酸逆转录酶抑制剂,可研究 HIV 和慢性乙型肝炎。
T16530 BF738735

Antiviral; PI4K Immunology/Inflammation; PI3K/Akt/mTOR signaling
BF738735 是有效的磷脂酰肌醇 4-激酶 IIIβ 抑制剂,IC50为 5.7 nM。
T60000 STING (WT/R232) activity regulator 126

STING Immunology/Inflammation
STING (WT/R232) activity regulator 126 是一种具有抗菌和抗病毒作用的 STING 调节剂。
T69188 Aloisine B

AloisineB

GSK-3; CDK Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells
Aloisine B (AloisineB) inhibited cyclin-dependent kinase and glycogen synthase kinase with IC50 values of 0.85 µM and 0.75 µM, respectively. Aloisine B has antiviral activity and can be used to study Alzheimer's, diabetes, HIV and Parkinson's.
T40276 GS-621763

SARS-CoV Microbiology/Virology
GS-621763 是具有口服活性的 GS-441524 前药,在小鼠体内具有抗SARS-CoV-2病毒活性。
T67807 Rociclovir PM

2-[(2-aminopurin-9-yl)methoxy]propane-1,3-diol

Antiviral Immunology/Inflammation
Rociclovir PM (2-[(2-aminopurin-9-yl)methoxy]propane-1,3-diol) 是一种具有抗病毒活性的化合物。
T29187 YM-53403

YM-53403是具有抗病毒活性,可有效抑制属于A 亚群和B 亚组的RSV 毒株的复制,可用来治疗呼吸道合胞病毒感染。
T0090 Moroxydine hydrochloride

盐酸吗啉胍,ABOB hydrochloride,病毒灵,Moroxydine HCl

Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Moroxydine hydrochloride (ABOB hydrochloride) 是一种合成的杂环双胍类抗病毒药物。 它具有抗病毒活性,有助于预防和治疗流感。
T28830 Sovaprevir

ACH 0141625,ACH0141625,ACH-0141625,ACH1625,ACH 1625,ACH-1625

HCV Protease Microbiology/Virology; Proteases/Proteasome
Sovaprevir 是一种非结构性3(NS3)蛋白酶抑制剂,有抗病毒活性,用于治疗 HCV 感染。
T16702 QL47

Virus Protease; BTK Angiogenesis; Microbiology/Virology; Tyrosine Kinase/Adaptors
QL47 是一种宿主靶向的小分子抗病毒剂,具有抗病毒活性,对登革热病毒和其他 RNA 病毒有抑制作用。QL47 可作为病毒翻译的抑制抑制剂和 BTK 的共价抑制剂,可用于研究淋巴瘤。
T5949 Dideoxyadenosine

2',3'-Dideoxyadenosine 是HIV 复制抑制剂,具有抗逆转录病毒活性和抗病毒的作用[1]。
T40293 GPS491

Antiviral; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
GPS491 具有抗病毒活性,通过改变 RNA 加工来抑制 HIV-1、腺病毒和冠状病毒复制。
T37340 N4-Acetylsulfamethoxazole

N-acetyl Sulfamethoxazole,醋磺胺甲噁唑

Others Others
N4-Acetylsulfamethoxazole 是磺胺甲恶唑的一种代谢物。Sulfamethoxazole 属于磺胺类抗菌素,可用于细菌感染。
T68015 Ruzasvir

MK8408,MK-8408,MK 8408

HCV Protease Microbiology/Virology; Proteases/Proteasome
Ruzasvir (MK-8408) 是一种新型有效的丙型肝炎病毒NS5A的泛基因型抑制剂,具有抗病毒活性。
T8371 ML188

Virus Protease; SARS-CoV Microbiology/Virology
ML188是一种选择性非共价 SARS-CoV3CLpro 抑制剂,具有抗病毒活性,IC50为 1.5 μM。
T68103 MK-6186

Reverse Transcriptase Microbiology/Virology
MK-6186 是一种新型非核苷类逆转录酶抑制剂,具有抗病毒活性,可用于研究病毒感染。
T11785 KT203

MAGL Metabolism
KT203 是一种具有选择性和高效性的 α/β 水解酶结构域 6 (ABHD6) 抑制剂,具有潜在的抗病毒和抗炎活性,可用于研究肺炎。
T9872 Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-

Others Others
Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-是一种用于抗病毒活性测定的化合物。
T9648 SIRT1-IN-1

Antiviral; Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation
SIRT1-IN-1 是一种选择性的 SIRT1 抑制剂,IC50 为 205 nM。 SIRT1-IN-1 是一种具有抗病毒活性的巨细胞病毒 (CMV) 抑制剂。
T67798 (2RS)-FPMPA

FPMPA

HIV Protease Microbiology/Virology; Proteases/Proteasome
(2RS)-FPMPA(FPMPA) 具有抗病毒活性,在感染SHIV(DH4R)的人MT12细胞的测得IC50 值为1.85μM。
T68103L Mk-6186 HCl

Mk-6186 HCl(1034474-19-5 Free base)

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
MK-6186 HCl,一种新型非核苷类逆转录酶抑制剂,具有抗病毒活性,可用于研究HIV。
T72051 LabMol-319

Virus Protease Microbiology/Virology
LabMol-319 是一种有效的寨卡病毒 (ZIKV) NS5 RdRp 抑制剂,具有抗病毒活性,可用于研究 ZIKV 病毒。
T9225 Vebicorvir

ABI-H0731

HBV Microbiology/Virology
Vebicorvir (ABI-H0731) 是一种乙型肝炎病毒核心蛋白的抑制剂,有抗病毒活性。
T16911 Sorivudine

BV-araU,索立夫定

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Sorivudine (BV-araU) 是口服有效的,嘧啶核苷抗代谢药物。它的抗病毒活性来自某些 DNA 病毒中存在的特定胸苷激酶选择性转化为核苷酸,从而反过来会干扰病毒 DNA 合成。
T26914L (R)-AZD 9639

Others Others
(R)-AZD 9639 是 AZD 9639 的 R型异构体。AZD 9639 是一种新型呼吸道合胞病毒(RSV)融合抑制剂,具有抗病毒活性。
T64396 Antiviral agent 38

Antiviral Immunology/Inflammation
Antiviral agent 38具有抗菌和抗病毒活性,可用来研究乙肝病毒。
T36113 Cobaltic Protoporphyrin IX chloride

Protoporphyrin IX cobaltic chloride

Autophagy Autophagy
Cobaltic Protoporphyrin IX chloride (CoPP)是一种有效的血红素加氧酶 1(HO-1)诱导剂,具有抗病毒活性,通过诱导 I 型 IFN 反应来抑制甲型流感病毒(IAV)感染。
T64091 (-)-JNJ-A07

Others Others
(-)-JNJ-A07 是一种具有选择性和高效性的登革热病毒 (DENV) 抑制剂(EC50:31 nM),具有抗病毒活性,可用于研究登革热病毒感染。
T23910 Cosalane

NSC 658586,NSC-658586,NSC 640067

HIV Protease Microbiology/Virology; Proteases/Proteasome
Cosalane (NSC 658586) 是一种 HIV 复制抑制剂,是人和小鼠趋化因子受体 7 (CCR7)信号传导的抑制剂,具有抗病毒活性,可阻断 CCR7 与其天然配体 CCL19 和 CCL21 结合。Cosalane 对多种 HIV-1 株系和 HIV-2 具有活性。
T16325 NITD008

7-Deaza-2'-C-acetylene-adenosine

Others Others
NITD008 (7-Deaza-2'-C-acetylene-adenosine) 是一种有效的和选择性的腺苷核苷抑制剂,是一种腺苷核苷类似物,具有广谱的抗病毒活性,抑制登革热病毒、动物杯状病毒和寨卡病毒。
T29955 AMC-01

AMC01,AMC 01

Antiviral; PERK Apoptosis; Immunology/Inflammation
AMC-01 具有潜在的抗病毒活,可通过丝氨酸残基 51 的磷酸化诱导 eIF2-α 失活,这种作用具有剂量和时间依赖性。AMC-01 可用来研究动脉粥样硬化和帕金森综合征。
T8328 STING agonist-1

G10

Virus Protease; STING Immunology/Inflammation; Microbiology/Virology
STING agonist-1 (G10)是一种人类特异性 STING 激动剂,可引发针对新兴甲病毒的抗病毒活性。它抑制甲病毒属 VEEV 复制,IC90值为 24.57 μM。
T77652 SARS-CoV-2 3CLpro-IN-20

Antiviral; SARS-CoV Immunology/Inflammation; Microbiology/Virology
SARS-CoV-2 3CLpro-IN-20 是一种共价的 SARS-CoV-2 3CLpro 抑制剂(IC50s: 0.43 μM,)。SARS-CoV-2 3CLpro-IN-20 具有潜在的抗病毒活性。

化合物

BVDV-IN-1
Cat.No: T9103
Synonym:
Target: DNA/RNA Synthesis
Inarigivir soproxil
Cat.No: T15573
Synonym: SB9200
Target: HCV Protease
5-Fluorocytidine
Cat.No: T8625
Synonym:
Target: Antiviral
Antiviral agent
Cat.No: T67904
Synonym:
Target: HBV
2-PADQZ hydrochloride
Cat.No: T19849L
Synonym: 2-PADQZ hydrochloride (60547-97-9 Free base)
Target: Antiviral, Influenza Virus
ABI-1968
Cat.No: T67785
Synonym:
Target:
R 61837
Cat.No: T26020
Synonym: R-61837,R61837
Target: Antiviral
Sotirimod
Cat.No: T16913
Synonym: R850,S-30594
Target: Virus Protease
Rociclovir
Cat.No: T67806
Synonym:
Target: Antiviral
Cefprozil
Cat.No: T1118L
Synonym: Cefprozilum,Cefprozilo,Cefzil,Brisoral,Cefprozil anhydrous
Target: Antibacterial, Antibiotic
BTA-9881
Cat.No: T26914
Synonym: BTA9881,AZD9639,AZD-9639,BTA 9881,MEDI-564
Target: RSV
DDG-39
Cat.No: T67797
Synonym: 1-(2,3-dideoxy-2-fluoropentofuranosyl)cytosine
Target: Antiviral, HBV, HIV Protease
Levovirin
Cat.No: T25702
Synonym: ICN 17261,L-Ribavirin,ICN-17261,ICN17261
Target:
IM-250
Cat.No: T80675
Synonym:
Target: Antiviral
SHEN26
Cat.No: T60014
Synonym:
Target: Antiviral
2’-beta-C-Methyl inosine
Cat.No: TNU0442
Synonym: 2'-C-Methylinosine
Target: Antiviral, DNA/RNA Synthesis
Abacavir sulfate
Cat.No: T6367
Synonym: Abacavir Hemisulfate,硫酸阿巴卡韦,1592U89,ABC sulfate,Ziagen
Target: Apoptosis, HIV Protease, Reverse Transcriptase
Tenofovir
Cat.No: T1649
Synonym: 替诺福韦,泰诺福韦,PMPA,TDF,GS 1278
Target: HBV, HIV Protease, Reverse Transcriptase
BF738735
Cat.No: T16530
Synonym:
Target: Antiviral, PI4K
STING (WT/R232) activity regulator 126
Cat.No: T60000
Synonym:
Target: STING
Aloisine B
Cat.No: T69188
Synonym: AloisineB
Target: GSK-3, CDK
GS-621763
Cat.No: T40276
Synonym:
Target: SARS-CoV
Rociclovir PM
Cat.No: T67807
Synonym: 2-[(2-aminopurin-9-yl)methoxy]propane-1,3-diol
Target: Antiviral
YM-53403
Cat.No: T29187
Synonym:
Target:
Moroxydine hydrochloride
Cat.No: T0090
Synonym: 盐酸吗啉胍,ABOB hydrochloride,病毒灵,Moroxydine HCl
Target: Antiviral, Influenza Virus
Sovaprevir
Cat.No: T28830
Synonym: ACH 0141625,ACH0141625,ACH-0141625,ACH1625,ACH 1625,ACH-1625
Target: HCV Protease
QL47
Cat.No: T16702
Synonym:
Target: Virus Protease, BTK
Dideoxyadenosine
Cat.No: T5949
Synonym:
Target:
GPS491
Cat.No: T40293
Synonym:
Target: Antiviral, HIV Protease
N4-Acetylsulfamethoxazole
Cat.No: T37340
Synonym: N-acetyl Sulfamethoxazole,醋磺胺甲噁唑
Target: Others
Ruzasvir
Cat.No: T68015
Synonym: MK8408,MK-8408,MK 8408
Target: HCV Protease
ML188
Cat.No: T8371
Synonym:
Target: Virus Protease, SARS-CoV
MK-6186
Cat.No: T68103
Synonym:
Target: Reverse Transcriptase
KT203
Cat.No: T11785
Synonym:
Target: MAGL
Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-
Cat.No: T9872
Synonym:
Target: Others
SIRT1-IN-1
Cat.No: T9648
Synonym:
Target: Antiviral, Sirtuin
(2RS)-FPMPA
Cat.No: T67798
Synonym: FPMPA
Target: HIV Protease
Mk-6186 HCl
Cat.No: T68103L
Synonym: Mk-6186 HCl(1034474-19-5 Free base)
Target: HIV Protease, Reverse Transcriptase
LabMol-319
Cat.No: T72051
Synonym:
Target: Virus Protease
Vebicorvir
Cat.No: T9225
Synonym: ABI-H0731
Target: HBV
Sorivudine
Cat.No: T16911
Synonym: BV-araU,索立夫定
Target: DNA/RNA Synthesis
(R)-AZD 9639
Cat.No: T26914L
Synonym:
Target: Others
Antiviral agent 38
Cat.No: T64396
Synonym:
Target: Antiviral
Cobaltic Protoporphyrin IX chloride
Cat.No: T36113
Synonym: Protoporphyrin IX cobaltic chloride
Target: Autophagy
(-)-JNJ-A07
Cat.No: T64091
Synonym:
Target: Others
Cosalane
Cat.No: T23910
Synonym: NSC 658586,NSC-658586,NSC 640067
Target: HIV Protease
NITD008
Cat.No: T16325
Synonym: 7-Deaza-2'-C-acetylene-adenosine
Target: Others
AMC-01
Cat.No: T29955
Synonym: AMC01,AMC 01
Target: Antiviral, PERK
STING agonist-1
Cat.No: T8328
Synonym: G10
Target: Virus Protease, STING
SARS-CoV-2 3CLpro-IN-20
Cat.No: T77652
Synonym:
Target: Antiviral, SARS-CoV
Cat. No. Product Name Target Signaling Pathways
T6S0923 Hypericin

Hypericine,金丝桃素,Cyclosan

Apoptosis; Antiviral; Influenza Virus; Tyrosine Kinases; Antibacterial; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Tyrosine Kinase/Adaptors
Hypericin (Cyclosan) 是贯叶连翘的提取物,有抗菌、抗病毒、抗肿瘤和抗抑郁作用。
T7972 Gallic aldehyde

3,4,5-三羟基苯甲醛,五倍子醛

HSV Microbiology/Virology
Gallic aldehyde 对 HSV-1 显示出有效的抗病毒活性。
T7994 3-Methoxyflavone

Antiviral Immunology/Inflammation
3-Methoxyflavone 是一种黄酮类化合物,分离自 Artemisia incanescens,具有抗病毒作用。
TN1693 Glabrone

Influenza Virus; PPAR DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Glabrone 是从甘草根中分离的一种异黄酮,可与 PPAR-γ 配体结合,具有抗流感活性。
TN5891 Seselin

Antiviral; Immunology/Inflammation related Immunology/Inflammation
Seselin 是来自 Plumbago zeylanica 的天然产品。 Seselin 具有抗炎和抗病毒活性。
T2S1158 4,5-Dicaffeoylquinic acid

3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C

Others; HBV; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) 是一种天然产物,有抗病毒、抗肝毒性活性。
T3345 Hederasaponin B

常春藤皂苷B,Eleutheroside M,刺五加叶中,Hederacoside B

Others; Virus Protease Microbiology/Virology; Others
Hederasaponin B (Hederacoside B) 是从Hedera helix 中分离的,有广谱抗病毒活性。
T2875 Angelicin

Isopsoralen,异补骨脂素

Apoptosis; Virus Protease; Antiviral Apoptosis; Immunology/Inflammation; Microbiology/Virology
Angelicin (Isopsoralen) 是一种三环芳烃天然产物,结构上跟补骨脂素有关,具有抗癌、抗炎、抗病毒等活性。
T6S2024 Harpagide

Antibacterial; Parasite Microbiology/Virology
Harpagide 是从Scrophularia cryptophila 中分离出来的一种鸢尾糖苷,具有抗炎和抗寄生虫活性,对T.b. rhodesiense 具有体外锥虫杀虫活性,IC50为 21 μg/mL,它对L. donovani 的IC50值为 2.0 μg/mL。
T8205 Norwogonin

5,7,8-Trihydroxyflavone,去甲汉黄芩素

Virus Protease Microbiology/Virology
Norwogonin (5,7,8-Trihydroxyflavone) 是从黄芩中分离出来的,对肠道病毒 71 具有抗病毒活性,IC50为 31.83 μg/ ml。
T25327 Didemnin B

NSC 325319,NSC325319,膜海鞘素B,NSC-325319,Didemnin-B

Antiviral Immunology/Inflammation
Didemnin B (Didemnin-B) 是一种从海洋金枪鱼 Tridemnin cyanophorum 中提取的脱脂肽,具有抗病毒和抗肿瘤活性。
T4593 ISOPIMPINELLIN

5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen

Antiviral; DNA/RNA Synthesis; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology
Isopimpinellin (4,9-Dimethoxypsoralen) 是从 Pimpinella saxifrage 根部分离得到的一种天然产物,具有抗病毒和抗利什曼病活性。
TN1453 Bruceantinol

Anti-infection Microbiology/Virology
Bruceantinol 是一种quassinol 化合物,分离自Brucea javanica 的 CH3OH 提取物。它能够将系统性寄主植物中灭活。有效的抑制浓度为 10 μM。
T4537 Cholic acid sodium

胆酸钠,[胆酸钠],SodiumCholate

HIV Protease; Endogenous Metabolite Metabolism; Microbiology/Virology; Proteases/Proteasome
Cholic acid sodium (SodiumCholate) 是肝脏中产生的主要胆汁酸,通常与牛磺酸或甘氨酸结合,有助于脂肪吸收和胆固醇排泄。
T75675 Nepasaikosaponin K

Antiviral Immunology/Inflammation
Nepasaikosaponin K 是一种从柴胡根中分离出来小分子化合物,具有抗流感和抗病毒活性,可用于研究病毒感染。
T6S2025 8-​O-​Acetylharpagide

8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide

Antibacterial Microbiology/Virology
8-O-Acetylharpagide 是从 Ajuga reptans 中分离得到的一种环烯醚萜,有抗肿瘤、抗病毒、抗菌和抗炎作用。它对豚鼠的离体平滑肌有生物活性。
T6742 2-Deoxy-D-glucose

2-Deoxy-D-arabino-hexose,2-deoxyglucose,D-Arabino-2-deoxyhexose,Ba 2758,D-2-脱氧葡萄糖,NSC 15193,2-DG,2-脱氧-D-葡萄糖

Apoptosis; Hexokinase; HSV Apoptosis; Metabolism; Microbiology/Virology
2-Deoxy-D-glucose (2-DG) 是葡萄糖的类似物,是一种糖酵解抑制剂。2-Deoxy-D-glucose 具有抗病毒活性,还具有抑制细胞增殖、诱导细胞凋亡的活性。
TN2315 Xanthopurpurin

茜草红素,1,3-二羥蒽醌,异茜草素

Platelet aggregation; Antifection Microbiology/Virology; Others
Xanthopurpurin 是分离自Rubia akane 根茎的蒽醌苷。Xanthopurpurin 主要对胶原诱导的血小板聚集有较强的抑制作用。
T10164 5,6-Dihydroxyindole

Dopamine lutine

Endogenous Metabolite Metabolism
5,6-Dihydroxyindole (Dopamine lutine) 是黑色素的前体,显示出广谱的抗菌,抗真菌,抗病毒,抗寄生虫活性。5,6-Dihydroxyindole 也显示出细胞毒性作用。
T1506 Vidarabine

Adenine Arabinoside,阿糖腺苷,9-β-D-Arabinofuranosyladenine,Vira-A,Arabinosyladenine,Ara-A

Nucleoside Antimetabolite/Analog; Tyrosine Kinases; DNA/RNA Synthesis; Antibiotic; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Tyrosine Kinase/Adaptors
Vidarabine (Adenine Arabinoside) 是从链霉菌分离的核苷类抗生素,能抗单纯性疱疹和水痘-带状疱疹病毒。它对 HSV-1 和 HSV-2 的 IC50值分别为 9.3 μg/ml 和 11.3 μg/ml。
T9715 Aplidine

SARS-CoV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Aplidine 是有效的eEF1A2(KD=80 nM) 靶向的抗癌药物。Aplidine 具有抗病毒活性,抑制SARS-CoV-2的 IC90为 0.88 nM。Aplidine 在多发性骨髓瘤,晚期癌症及 COVID-19 领域有研究的价值。
T4S0999 (2S)-Isoxanthohumol

Isoxanthohumol,(2S)-异黄腐酚,异黄腐醇

Virus Protease; HSV Microbiology/Virology
(2S)-Isoxanthohumol 是一种由啤酒花原异戊烯基二氢黄酮 Isoxanthohumol 的微生物转化代谢物。
T7054 N-Benzoyl-(2R,3S)-3-phenylisoserine

N-苯甲酰基-(2R,3S)-3-苯基异丝氨酸,taxol side chain

Antiviral Immunology/Inflammation
N-Benzoyl-(2R,3S)-3-phenylisoserine (taxol side chain) 是一种制备用于研究结合位点位置的强效抗癌药物紫杉醇的中间体。 它显示出细胞毒性、抗病毒和免疫调节活性。
TN2755 2-Desoxy-4-epi-pulchellin

Anti-infection Microbiology/Virology
2-Desoxy-4-epi-pulchellin 是分离自 Polygonum hydropiper 的二氯甲烷可溶部分的一种化合物。
T75643 Isoxanthohumol

HSV Microbiology/Virology
Isoxanthohumol 是一种从啤酒花和啤酒中提取的一种前黄酮类化合物,对几种人类癌细胞株具有抗增殖活性。Isoxanthohumol对肿瘤细胞肺转移灶的转移或侵袭有抑制作用。Isoxanthohumol具有抗病毒活性,对疱疹病毒(HSV1和HSV2)和牛病毒性腹泻病毒(BVDV)具有抑制作用。
T0884 1-Docosanol

Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol

Antifection; HSV Microbiology/Virology
1-Docosanol (Behenic alcohol) 是一种具有抗病毒活性的饱和 22 碳脂肪醇,局部用于治疗复发性单纯性唇疱疹发作并缓解相关疼痛并可能有助于更快地治愈疮。
TN2331 Eleutheroside B1

刺五加苷B1

Influenza Virus Microbiology/Virology
Eleutheroside B1是具有广谱抗人流感病毒的一种香豆素。它抑制多种趋化因子基因和流感病毒核蛋白基因的 mRNA 表达。它具有抗病毒、抗流感和抗炎活性,且细胞毒性小。
T38251 L-Uridine

Nucleoside Antimetabolite/Analog; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
L-Uridine 是从Polyporaceae fungus Poria cocos (Schw.)分离得到的正常 RNA 成分中的 D-尿苷的对映异构体,属于一种核苷,可充当核苷磷酸转移酶的磷酸受体。L-Uridine 具有潜在的抗病毒活性。
T4S1335 Daphnoretin

Dephnoretin,西瑞香素,Thymelol

Influenza Virus; Caspase; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
Daphnoretin (Thymelol) 是从了哥王中提取得到的一种天然产物,具有抗癌和抗病毒活性。它通过在 G2/M 期连续阻断细胞并激活 caspase-3 通路导致 HOS 细胞死亡。
T5S2059 Glaucine

Calcium Channel; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; PDE GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Glaucine 是从海罂粟中分离的一种生物碱,具有镇咳、抗炎和支气管扩张作用。它是具有口服活性的磷酸二酯酶 4 选择性抑制剂。它还是非选择性的 α-肾上腺素受体拮抗剂,具有抗氧化和抗病毒活性。
T6S2391 L-Chicoric Acid

(-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸,是一种选择性可逆的 HIV-1 整合酶抑制剂,IC50约为 100 nM。它还可抑制 HIV-1 复制。
T3795 Corilagin

Apoptosis; TLR; Reverse Transcriptase; Antibacterial; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology
Corilagin 是一种鞣酸,有抑制 RNA 肿瘤病毒逆转录酶的活性。它抑制金黄色葡萄球菌的生长,MIC 为 25 μg/mL。它有抗肿瘤活性,可用于肝癌和卵巢癌。
T2S1865 Octyl gallate

Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯

Antioxidant; Influenza Virus; Reactive Oxygen Species; Antibacterial; Antifungal; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) 具有抗菌、抗氧化作用,有选择性和敏感性的荧光特性,广泛用作食品添加剂。它对 HSV-1,水泡性口炎病毒和脊髓灰质炎病毒有显著的抗病毒作用。
TN6066 1-Hydroxyacridone

1-Hydroxyacridone has potential antiviral activity.
TN2395 Epirengynic acid

Antiviral Immunology/Inflammation
Epirengynic acid has antiviral activity against RSV
T12995 Squalamine

MSI-1256,角鲨胺

Others Others
Squalamine is an aminosterol compound, with potent broad spectrum antiviral activity.
TN6420 Sikokianin A

Sikokianin A shows in vitro antiviral activity against HBsAg secretion.
TN3713 Corymbosin

Antifection Microbiology/Virology
Corymbosin shows significant antiviral activity.
TN2321 Yadanzioside L

Antifection Microbiology/Virology
Yadanzioside L shows strong antiviral activity.
TN5267 Yadanzioside I

Antifection Microbiology/Virology
Yadanzioside I shows strong antiviral activity.
TN2417 Furomollugin

5-羟基萘并[1,2-B]呋喃-4-甲酸甲酯,呋喃大叶茜草素

Antifection Microbiology/Virology
Furomollugin has antiviral activity, it can strongly suppress the secretion of hepatitis B surface antigen (HBsAg), with IC50 = 2.0 micrograms/mL, in human hepatoma Hep3B cells.
TN2220 Sophoranol

槐醇,(+)-Sophoranol

HBV Microbiology/Virology
(+)-Sophoranol exhibits antiviral activity against the Coxsackie virus B3. It also shows potent anti-HBV activity with an inhibitory potency against HBsAg secretion and against HBeAg secretion.
TN4932 Sageone

PARP; Akt; Caspase; Antifection Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Sageone represents a promising anticancer agent against gastric cancer that warrants further study, it synergizes with cisplatin cytotoxicity in SNU-1 human gastric cancer cells.Sageone also shows antiviral activity.
T25789 Melianone

NSC 302037,NSC-302037,NSC302037

Melianone exhibits antiviral activity (EC50s: 3-11μM) against three important human pathogens, belonging to the Flaviviridae family, West Nile virus, Dengue virus, and Yellow Fever virus.
T8263 3,4'-Dihydroxyflavone

Influenza Virus Microbiology/Virology
3,4'-Dihydroxyflavone 是一种口服活性黄酮类化合物,具有抗甲型流感病毒的抗病毒活性。
TN5717 6'-O-Galloylsalidroside

Antiviral; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
6'-O-Galloylsalidroside 具有抗病毒活性,对HIV 具有抑制作用。
TN1843 Kushenol K

PDE; HSV Metabolism; Microbiology/Virology
Kushenol K is a potent and Selective Inhibitor of cGMP Phosphodiesterase 5, it also has inhibitory effects on diacylglycerol acyltransferase (DGAT). Kushenol K shows weak antiviral activity against Herpes simplex virus types I and II.
TN4456 Lucidadiol

AChR; HSV Microbiology/Virology; Neuroscience
Lucidadiol exhibits butyrylcholinesterase-inhibitory activity at concentrations up to 200 uM, it also possesses inhibitory activity against acetylcholinesterase (AChE) with the percentage inhibition at 100 uM. Lucidadiol shows antiviral activity against i
TN1632 Euparin

Antifection Microbiology/Virology
Euparin exhibits a moderate antioxidant activity, it also exhibits antifungal activity against Trichophyton mentagrophytes. Euparin has antiviral activity, it exerts its effect during the early events of the replication cycle, from the virus adsorption to
T3930 Taraxerol acetate

醋酸蒲公英霜,Taraxeryl acetate

Phosphatase; HSV Metabolism; Microbiology/Virology
Taraxeryl acetate shows the significant antiviral activity against herpes simplex virus (type II). It has less effect on cell cycle arrest and apoptosis of AGS cells than taraxerol. A. roxburghiana has antidiabetic activity, could be attributed due to PTP
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天然产物

Hypericin
Cat.No: T6S0923
Synonym: Hypericine,金丝桃素,Cyclosan
Target: Apoptosis, Antiviral, Influenza Virus, Tyrosine Kinases, Antibacterial, PKC
Gallic aldehyde
Cat.No: T7972
Synonym: 3,4,5-三羟基苯甲醛,五倍子醛
Target: HSV
3-Methoxyflavone
Cat.No: T7994
Synonym:
Target: Antiviral
Glabrone
Cat.No: TN1693
Synonym:
Target: Influenza Virus, PPAR
Seselin
Cat.No: TN5891
Synonym:
Target: Antiviral, Immunology/Inflammation related
4,5-Dicaffeoylquinic acid
Cat.No: T2S1158
Synonym: 3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C
Target: Others, HBV, Endogenous Metabolite
Hederasaponin B
Cat.No: T3345
Synonym: 常春藤皂苷B,Eleutheroside M,刺五加叶中,Hederacoside B
Target: Others, Virus Protease
Angelicin
Cat.No: T2875
Synonym: Isopsoralen,异补骨脂素
Target: Apoptosis, Virus Protease, Antiviral
Harpagide
Cat.No: T6S2024
Synonym:
Target: Antibacterial, Parasite
Norwogonin
Cat.No: T8205
Synonym: 5,7,8-Trihydroxyflavone,去甲汉黄芩素
Target: Virus Protease
Didemnin B
Cat.No: T25327
Synonym: NSC 325319,NSC325319,膜海鞘素B,NSC-325319,Didemnin-B
Target: Antiviral
ISOPIMPINELLIN
Cat.No: T4593
Synonym: 5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen
Target: Antiviral, DNA/RNA Synthesis, Parasite
Bruceantinol
Cat.No: TN1453
Synonym:
Target: Anti-infection
Cholic acid sodium
Cat.No: T4537
Synonym: 胆酸钠,[胆酸钠],SodiumCholate
Target: HIV Protease, Endogenous Metabolite
Nepasaikosaponin K
Cat.No: T75675
Synonym:
Target: Antiviral
8-​O-​Acetylharpagide
Cat.No: T6S2025
Synonym: 8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide
Target: Antibacterial
2-Deoxy-D-glucose
Cat.No: T6742
Synonym: 2-Deoxy-D-arabino-hexose,2-deoxyglucose,D-Arabino-2-deoxyhexose,Ba 2758,D-2-脱氧葡萄糖,NSC 15193,2-DG,2-脱氧-D-葡萄糖
Target: Apoptosis, Hexokinase, HSV
Xanthopurpurin
Cat.No: TN2315
Synonym: 茜草红素,1,3-二羥蒽醌,异茜草素
Target: Platelet aggregation, Antifection
5,6-Dihydroxyindole
Cat.No: T10164
Synonym: Dopamine lutine
Target: Endogenous Metabolite
Vidarabine
Cat.No: T1506
Synonym: Adenine Arabinoside,阿糖腺苷,9-β-D-Arabinofuranosyladenine,Vira-A,Arabinosyladenine,Ara-A
Target: Nucleoside Antimetabolite/Analog, Tyrosine Kinases, DNA/RNA Synthesis, Antibiotic, HSV
Aplidine
Cat.No: T9715
Synonym:
Target: SARS-CoV, DNA/RNA Synthesis
(2S)-Isoxanthohumol
Cat.No: T4S0999
Synonym: Isoxanthohumol,(2S)-异黄腐酚,异黄腐醇
Target: Virus Protease, HSV
N-Benzoyl-(2R,3S)-3-phenylisoserine
Cat.No: T7054
Synonym: N-苯甲酰基-(2R,3S)-3-苯基异丝氨酸,taxol side chain
Target: Antiviral
2-Desoxy-4-epi-pulchellin
Cat.No: TN2755
Synonym:
Target: Anti-infection
Isoxanthohumol
Cat.No: T75643
Synonym:
Target: HSV
1-Docosanol
Cat.No: T0884
Synonym: Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol
Target: Antifection, HSV
Eleutheroside B1
Cat.No: TN2331
Synonym: 刺五加苷B1
Target: Influenza Virus
L-Uridine
Cat.No: T38251
Synonym:
Target: Nucleoside Antimetabolite/Analog, Antibiotic
Daphnoretin
Cat.No: T4S1335
Synonym: Dephnoretin,西瑞香素,Thymelol
Target: Influenza Virus, Caspase, PKC
Glaucine
Cat.No: T5S2059
Synonym:
Target: Calcium Channel, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, PDE
L-Chicoric Acid
Cat.No: T6S2391
Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸
Target: Others, HIV Protease
Corilagin
Cat.No: T3795
Synonym:
Target: Apoptosis, TLR, Reverse Transcriptase, Antibacterial, Autophagy
Octyl gallate
Cat.No: T2S1865
Synonym: Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯
Target: Antioxidant, Influenza Virus, Reactive Oxygen Species, Antibacterial, Antifungal, HSV
1-Hydroxyacridone
Cat.No: TN6066
Synonym:
Target:
Epirengynic acid
Cat.No: TN2395
Synonym:
Target: Antiviral
Squalamine
Cat.No: T12995
Synonym: MSI-1256,角鲨胺
Target: Others
Sikokianin A
Cat.No: TN6420
Synonym:
Target:
Corymbosin
Cat.No: TN3713
Synonym:
Target: Antifection
Yadanzioside L
Cat.No: TN2321
Synonym:
Target: Antifection
Yadanzioside I
Cat.No: TN5267
Synonym:
Target: Antifection
Furomollugin
Cat.No: TN2417
Synonym: 5-羟基萘并[1,2-B]呋喃-4-甲酸甲酯,呋喃大叶茜草素
Target: Antifection
Sophoranol
Cat.No: TN2220
Synonym: 槐醇,(+)-Sophoranol
Target: HBV
Sageone
Cat.No: TN4932
Synonym:
Target: PARP, Akt, Caspase, Antifection
Melianone
Cat.No: T25789
Synonym: NSC 302037,NSC-302037,NSC302037
Target:
3,4'-Dihydroxyflavone
Cat.No: T8263
Synonym:
Target: Influenza Virus
6'-O-Galloylsalidroside
Cat.No: TN5717
Synonym:
Target: Antiviral, HIV Protease
Kushenol K
Cat.No: TN1843
Synonym:
Target: PDE, HSV
Lucidadiol
Cat.No: TN4456
Synonym:
Target: AChR, HSV
Euparin
Cat.No: TN1632
Synonym:
Target: Antifection
Taraxerol acetate
Cat.No: T3930
Synonym: 醋酸蒲公英霜,Taraxeryl acetate
Target: Phosphatase, HSV
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